Publications

Ion mobility mass spectrometry unveils conformational effects of drug lead EPI-001 on the intrinsically disordered N-terminal domain of the Androgen Receptor

Ahmed Ikhlas M M, Rofe Adam, Henry Martyn C, West Eric, Jamieson Craig, McEwan Iain J, Beveridge Rebecca

Protein Science Vol 34 (2025)

https://doi.org/10.1002/pro.5254

One-pot oxidative amidation of aldehydes via the generation of nitrile imine intermediates

Henry Martyn C, Minty Laura, Kwok Alexander C W, Elwood Jessica M L, Foulis Adam J, Pettinger Jonathan, Jamieson Craig

Journal of Organic Chemistry Vol 89, pp. 7913-7926 (2024)

https://doi.org/10.1021/acs.joc.4c00575

Synthesis and evaluation of small molecule inhibitors of the androgen receptor N-terminal domain

Henry Martyn C, Riley Christopher M, Hunter Irene, Elwood Jessica M L, Lopez-Fernandez J Daniel, Minty Laura, Coe Diane M, McEwan Iain J, Jamieson Craig

ACS Medicinal Chemistry Letters Vol 14, pp. 1800-1806 (2023)

https://doi.org/10.1021/acsmedchemlett.3c00426

Current and emerging approaches to noncompetitive AR inhibition

Riley Christopher M, Elwood Jessica M L, Henry Martyn C, Hunter Irene, Lopez-Fernandez J Daniel, McEwan Iain J, Jamieson Craig

Medicinal Research Reviews Vol 43, pp. 1701-1747 (2023)

https://doi.org/10.1002/med.21961

Multigram-scale synthesis of a gem-difluoro-substituted 4,5,6,7-tetrahydrobenzo[c]thiophen-4-one heterocycle via oxidative chlorination and radical Smiles rearrangement

Henry Martyn C, Anderson Jack Q, Jamieson Craig

Synlett Vol 34 (2023)

https://doi.org/10.1055/a-2153-7341

Functionalized tetrazoles as latent active esters in the synthesis of amide bonds

Elwood Jessica M L, Henry Martyn C, Lopez-Fernandez J Daniel, Mowat Jenna M, Boyle Mhairi, Buist Benjamin, Livingstone Keith, Jamieson Craig

Organic Letters Vol 24, pp. 9491-9496 (2022)

https://doi.org/10.1021/acs.orglett.2c03971

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